Tolvaptan is a selective and competitive arginine vasopressin receptor 2 antagonist. Vasopressin acts on the V2 receptors found in the
Vasopressin antagonists are drugs that bind to vasopressin receptors (V1A, V1B and V2) and block the action of vasopressin (antidiuretic hormone, ADH), which is a hormone released by the pituitary gland.
Antidiuretic Hormone Receptor Antagonists ; Tolvaptan Vasopressin V1a receptor, target ; Satavaptan Vasopressin V2 receptor, target ; Balovaptan Vasopressin
Serotonin receptor 1A agonist/serotonin receptor 2A antagonist: flibanserin. Vasopressin receptor antagonists: tolvaptan. ➢ Drugs that are strong CYP3A
The recent emergence of vasopressin receptor antagonists provides a class of drugs that target the primary pathophysiological mechanism, namely vasopressin
Vasopressin antagonists are drugs that bind to vasopressin receptors (V1A, V1B and V2) and block the action of vasopressin (antidiuretic hormone, ADH).
Therapeutic potential of vasopressin receptor antagonists. Drugs. 2024; . PUBMED
What are Vasopressin antagonists? Vasopressin antagonists are drugs that bind to vasopressin receptors (V1A, V1B and V2) and block the action of vasopressin (
A vasopressin receptor antagonist (VRA) is an agent that interferes with action at the vasopressin receptors. Most commonly VRAs are used in the treatment
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